RS 67333 hydrochloride

CAS No. 168986-60-5

RS 67333 hydrochloride ( RS 67333 HCl; RS 67333 (hydrochloride) )

Catalog No. M27698 CAS No. 168986-60-5

potent and highly selective 5-HT4 partial agonist.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
5MG 65 Get Quote
10MG 110 Get Quote
25MG 259 Get Quote
50MG 407 Get Quote
100MG 599 Get Quote
200MG Get Quote Get Quote
500MG Get Quote Get Quote
1G Get Quote Get Quote

Biological Information

  • Product Name
    RS 67333 hydrochloride
  • Note
    Research use only, not for human use.
  • Brief Description
    potent and highly selective 5-HT4 partial agonist.
  • Description
    potent and highly selective 5-HT4 partial agonist.(In Vitro):RS 67333 hydrochloride exhibits affinities for the sigma 1 (pKi = 8.9) and sigma 2 (pKi = 8.0) binding sites. At the 5-HT4 receptor mediating relaxation of the carbachol-precontracted oesophagus, RS 67333 hydrochloride acts as a potent (pEC50 of 8.4), partial agonists (intrinsic activities, with respect to 5-HT is 0.5) with respect to 5-HT .
  • Synonyms
    RS 67333 HCl; RS 67333 (hydrochloride)
  • Pathway
    Others
  • Target
    Other Targets
  • Recptor
    c-Fgr;Lyn;Hck;Apoptosis
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    168986-60-5
  • Formula Weight
    389.4
  • Molecular Formula
    C19H30Cl2N2O2
  • Purity
    >98% (HPLC)
  • Solubility
    ——
  • SMILES
    Cl.CCCCN1CCC(CCC(=O)c2cc(Cl)c(N)cc2OC)CC1
  • Chemical Name
    ——

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1.Weir MC, et al. Selective Inhibition of the Myeloid Src-Family Kinase Fgr Potently Suppresses AML Cell Growth in Vitro and in Vivo. ACS Chem Biol. 2018 Jun 15;13(6):1551-1559.
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